1H-Benzimidazole-5-carboxamidine derivatives: design, synthesis, molecular docking, DFT and antimicrobial studies
Author:
Affiliation:
1. Erciyes University
2. Faculty of Pharmacy
3. Department of Pharmaceutical Chemistry
4. Kayseri
5. Turkey
6. Ankara University
7. Ankara
8. Trakya University
9. Department of Pharmaceutical Microbiology
10. Edirne
Abstract
15 new 1H-benzimidazole-5-carboxamidine derivatives were synthesized, their antimicrobial effects were evaluated, and molecular docking and DFT studies were performed.
Funder
Türkiye Bilimsel ve Teknolojik Araştirma Kurumu
Publisher
Royal Society of Chemistry (RSC)
Subject
Materials Chemistry,General Chemistry,Catalysis
Link
http://pubs.rsc.org/en/content/articlepdf/2020/NJ/D0NJ01899F
Reference79 articles.
1. Molecular mechanisms of antibiotic resistance
2. Bad Bugs, No Drugs: No ESKAPE! An Update from the Infectious Diseases Society of America
3. W. Kaplan and R.Laing , Priority medicines for Europe and the world , World Health Organization , Geneva , 2004
4. The role of vaccines in preventing bacterial antimicrobial resistance
5. blaI and blaR1 regulate beta-lactamase and PBP 2a production in methicillin-resistant Staphylococcus aureus
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