Regioselective “hydroamination” of alk-3-ynones with non-symmetrical o-phenylenediamines. Synthesis of diversely substituted 3H-1,5-benzodiazepines via (Z)-3-amino-2-alkenones
Author:
Affiliation:
1. Department of Chemistry
2. Oakland University
3. Rochester
4. USA
5. University of Massachusetts Boston
6. Boston
7. Eastern Illinois University
8. Charleston
9. Centre of Molecular and Macromolecular Studies
Abstract
Reaction of alk-3-yn-1-ones with non-symmetricalo-phenylenediamines provides an effective method with high atom economy for the synthesis of diversely substituted 1,5-benzodiazepines and conjugated enaminones.
Funder
American Chemical Society Petroleum Research Fund
National Science Foundation
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemical Engineering,General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2016/RA/C6RA24291J
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3. Construction of the 1,5-Benzodiazepine Skeleton from o-Phenylendiamine and Propargylic Alcohols via a Domino Gold-Catalyzed Hydroamination/Cyclization Process
4. Facile synthesis of both perfluoroalkyl and phosphonate groups substituted trans-1,5-benzodiazepine and its derivatives via a one-pot catalyst-free process
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