A quick access to CF<sub>3</sub>-containing functionalized benzofuranyl, benzothiophene and indolyl heterocycles under catalyst-free conditions-Reference-Cited by-同舟云学术

A quick access to CF₃-containing functionalized benzofuranyl, benzothiophene and indolyl heterocycles under catalyst-free conditions

Published:2024 Issue:70 Volume:60 Page:9376-9379
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Kazi Ayazoddin Aunoddin¹²,Manjuladevi Nadimpalli¹,Kumar Salla Suresh¹²,Sharma Anamika²³^ORCID,Singh L Ravithej¹²^ORCID

Affiliation:

1. Fluoro-Agrochemicals Division, CSIR-Indian Institute of Chemical Technology, Hyderabad-500 007, India

2. Chemical Sciences Division, Academy of Scientific and Innovative Research, Ghaziabad-201 002, India

3. Department of Natural Products and Medicinal Chemistry, CSIR-Indian Institute of Chemical Technology, Hyderabad-500 007, India

Abstract

2-BTP as a benign CF3 synthon, a catalyst-free one-pot synthetic protocol is presented for the preparation of trifluoromethyl containing benzofuran, indolin, and benzothiophene derivatives using readily available aromatic aldehydes and ketones.

Funder

Council of Scientific and Industrial Research, India

Department of Science and Technology, Ministry of Science and Technology, India

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/CC/D4CC02395A

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