Experimental and computational evidence for KOt-Bu-promoted synthesis of oxopyrazino[1,2-a]indoles-Reference-Cited by-同舟云学术

Experimental and computational evidence for KOt-Bu-promoted synthesis of oxopyrazino[1,2-a]indoles

Published:2015 Issue:123 Volume:5 Page:101353-101361
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Mahdavi Mohammad¹²³⁴⁵,Hassanzadeh-Soureshjan Rasoul⁶⁷⁸⁴⁵,Saeedi Mina⁹¹⁰³⁴⁵,Ariafard Alireza¹¹¹²¹³¹⁴¹⁵,BabaAhmadi Rasool¹⁶¹⁷¹⁸¹⁹²⁰,Ranjbar Parviz Rashidi⁶⁷⁸⁴⁵,Shafiee Abbas¹²³⁴⁵

Affiliation:

1. Department of Medicinal Chemistry

2. Faculty of Pharmacy and Pharmaceutical Sciences Research Center

3. Tehran University of Medical Sciences

4. Tehran

5. Iran

6. School of Chemistry

7. University College of Science

8. University of Tehran

9. Medicinal Plants Research Center

10. Faculty of Pharmacy

11. School of Physical Sciences (Chemistry)

12. University of Tasmania

13. Private Bag 75

14. Hobart TAS 7001

15. Australia

16. Department of Chemistry

17. Faculty of Science

18. Central Tehran Branch

19. Islamic Azad University

20. Shahrak Gharb

Abstract

Metal-free intramolecular hydroamination of some Ugi adducts in the presence of KOt-Bu in DMF at room temperature led to the formation of novel oxopyrazino[1,2-a]indole derivatives.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA17056G

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