Involvement of covalent interactions in the mode of action of PPARβ/δ antagonists-Reference-Cited by-同舟云学术

Involvement of covalent interactions in the mode of action of PPARβ/δ antagonists

Published:2015 Issue:93 Volume:5 Page:76483-76490
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Kaupang Åsmund¹²³⁴⁵,Hildonen Siri¹²³⁴⁵,Halvorsen Trine G.¹²³⁴⁵,Mortén Magnus⁶³⁷⁵,Vik Anders¹²³⁴⁵,Hansen Trond Vidar¹²³⁴⁵

Affiliation:

1. Department of Pharmaceutical Chemistry

2. School of Pharmacy

3. University of Oslo

4. 0316 Oslo

5. Norway

6. Department of Chemistry

7. 0315 Oslo

Abstract

Investigations on the mode of action of several different chemical modulators of the peroxisome proliferator-activated receptor β/δ (PPARβ/δ) have been reported using MS and NMR experiments.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA15707B

Reference82 articles.

1. Regulation of Skeletal Muscle Physiology and Metabolism by Peroxisome Proliferator-Activated Receptor δ

2. The contrasting roles of PPARδ and PPARγ in regulating the metabolic switch between oxidation and storage of fats in white adipose tissue

3. Transcriptional Repression of Atherogenic Inflammation: Modulation by PPARδ

4. PPARδ Enhances Keratinocyte Proliferation in Psoriasis and Induces Heparin-Binding EGF-Like Growth Factor

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