Room temperature N-arylation of amino acids and peptides using copper(i) and β-diketone
Author:
Affiliation:
1. Department of Medicinal Chemistry
2. National Institute of Pharmaceutical Education and Research
3. S. A. S. Nagar
4. India
Abstract
A mild and efficient Cu-catalyzed procedure for the N-arylation of zwitterionic amino acids, amino acid esters and peptides is described.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB00288E
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5. J. P. Greenstein and M.Wintz, Chemistry of the amino acids, John Wiley & Sons Inc., New York, 1961, vol. 1, p. 569
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