Affiliation:
1. Department of Chemistry and Biomolecular Sciences, University of Ottawa, Ottawa, Ontario K1N 6N5, Canada
Abstract
Our investigation of small, irreversible TG2 inhibitors identifies key components that confer enhanced efficiency, and reveals potential discrepancies in the use of current crystallographic models for predicting inhibitor potency.
Funder
Canadian Institutes of Health Research
Natural Sciences and Engineering Research Council of Canada
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Biochemistry
Cited by
8 articles.
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