Polysubstituted 3-trifluoromethylpyrazoles: regioselective (3 + 2)-cycloaddition of trifluoroacetonitrile imines with enol ethers and functional group transformations-Reference-Cited by-同舟云学术

Polysubstituted 3-trifluoromethylpyrazoles: regioselective (3 + 2)-cycloaddition of trifluoroacetonitrile imines with enol ethers and functional group transformations

Published:2018 Issue:8 Volume:16 Page:1252-1257
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Utecht Greta¹²³⁴,Fruziński Andrzej⁵⁶⁷⁴,Jasiński Marcin¹²³⁴^ORCID

Affiliation:

1. Faculty of Chemistry

2. University of Łódź

3. 91-403 Łódź

4. Poland

5. Institute of General and Ecological Chemistry

6. Łódź University of Technology

7. 90-924 Łódź

Abstract

Enol ethers were used as synthetic equivalents of alkynes in the reaction with in situ generated trifluoroacetonitrile imines to give 3-trifluoromethylpyrazoles in a fully regioselective manner.

Funder

Narodowe Centrum Nauki

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/OB/C7OB03126B

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