Synthesis of fluoro-benzoxazepines via an I(<scp>iii</scp>)/BF3·Et2O-enabled 1,2-aryl migration/fluorination cascade-Reference-Cited by-同舟云学术

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Synthesis of fluoro-benzoxazepines via an I(iii)/BF₃·Et₂O-enabled 1,2-aryl migration/fluorination cascade

Published:2024 Issue:17 Volume:11 Page:4805-4811
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

He Jiaxin¹,Shi Haofeng¹,Wu Jialiang¹,Xiao Dan¹,Yang Kaiyue¹,Sun Yuli¹,Du Yunfei¹^ORCID

Affiliation:

1. Tianjin Key Laboratory for Modern Drug Delivery & High-Efficiency, School of Pharmaceutical Science and Technology, Faculty of Medicine, Tianjin University, Tianjin 300072, China

Abstract

A metal-free method for constructing benzoxazepine backbone lies in an exclusive 1,2-aryl migration/ fluorination cascade process, which is enabled by a phenyliodine(iii) diacetate (PIDA)/BF3·Et2O reagents system.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/QO/D4QO00715H

Reference52 articles.

1. Synthesis and Biological Activities of Substituted Benzoxazepine: A Review

2. One-Pot Synthesis of Diverse Collections of Benzoxazepine and Indolopyrazine Fused to Heterocyclic Systems

3. A Synthetic Overview of Benzoxazines and Benzoxazepines as Anticancer Agents

4. Revisiting loxapine: a systematic review

5. Amoxapine

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