A general metal free approach to α-ketoamides via oxidative amidation–diketonization of terminal alkynes-Reference-Cited by-同舟云学术

A general metal free approach to α-ketoamides via oxidative amidation–diketonization of terminal alkynes

Published:2014 Issue:67 Volume:50 Page:9533-9535
ISSN:1359-7345
Container-title:Chem. Commun.
language:en
Short-container-title:Chem. Commun.

Author:

Deshidi Ramesh¹²³⁴,Kumar Manjeet¹²³⁴,Devari Shekaraiah¹²³⁴,Shah Bhahwal Ali¹²³⁴

Affiliation:

1. Academy of Scientific and Innovative Research (AcSIR)

2. Natural Product Microbes

3. CSIR-Indian Institute of Integrative Medicine

4. Jammu-Tawi, India

Abstract

A metal free catalytic system employing TMSOTf/I₂/DMSO for the oxidative amidation–diketonization of terminal alkynes, in order to produce a wide variety of α-ketoamides, has been developed.

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2014/CC/C4CC03783A

Reference34 articles.

1. Convergent Synthesis of α-Ketoamide Inhibitors of Pin1

2. Novel Peptidyl α-Keto Amide Inhibitors of Calpains and Other Cysteine Proteases

3. P2-achiral, P'-extended α-ketoamide inhibitors of calpain I

4. Fluoresceinated FKBP12 ligands for a high-throughput fluorescence polarization assay

5. Synthesis of di- and tripeptide analogues containing α-ketoamide as a new core structure for inhibition of HIV-1 protease

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