Synthesis of 3-aryl-2-aminoquinolines: palladium-catalyzed cascade reactions of gem-dibromovinylanilines with tert-butyl isocyanide and arylboronic acids-Reference-Cited by-同舟云学术

Synthesis of 3-aryl-2-aminoquinolines: palladium-catalyzed cascade reactions of gem-dibromovinylanilines with tert-butyl isocyanide and arylboronic acids

Published:2014 Issue:72 Volume:4 Page:38258-38262
ISSN:2046-2069
Container-title:RSC Adv.
language:en
Short-container-title:RSC Adv.

Author:

Hu Langxi¹²³⁴,Gui Weijun¹²³⁴,Liu Zichen⁵⁶⁷,Jiang Baishan¹²³⁴^ORCID

Affiliation:

1. Institute of Chemical Biology

2. Guangzhou Institutes of Biomedicine and Health

3. Chinese Academy of Sciences

4. Guangzhou 510530, China

5. Shenzhen University Health Science Center

6. Shenzhen University

7. China

Abstract

A three-component cascade reaction involving gem-dibromovinylanilines, tert-butyl isocyanide and arylboronic acids for the efficient synthesis of 3-aryl-2-aminoquinolines has been developed.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/RA/C4RA05670A

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4. 2,4-Diamino-6,7-dimethoxyquinoline derivatives as .alpha.1-adrenoceptor antagonists and antihypertensive agents

5. Development of CXCR3 antagonists. Part 4: Discovery of 2-amino-(4-tropinyl)quinolines

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