Synthesis of 2-substituted 3-chlorobenzofurans via TMSCl-mediated nucleophilic annulation of isatin-derived propargylic alcohols-Reference-Cited by-同舟云学术

Synthesis of 2-substituted 3-chlorobenzofurans via TMSCl-mediated nucleophilic annulation of isatin-derived propargylic alcohols

Published:2018 Issue:33 Volume:16 Page:6133-6139
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Sun Zhou¹²³⁴,Xiang Kuirong¹²³⁴,Tao Hua⁵⁶⁷,Guo Liqun¹²³⁴,Li Ying¹²³⁴^ORCID

Affiliation:

1. State Key Laboratory of Applied Organic Chemistry & College of Chemistry and Chemical Engineering

2. Lanzhou University

3. Lanzhou

4. P. R. of China

5. Northwest Institute of Eco-Environmental and Resorce

6. CAS

7. China

Abstract

A TMSCl-mediated cascade annulation of isatin-derived propargylic alcohols has been developed for the facile synthesis of 2-substituted 3-chlorobenzofurans.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/OB/C8OB01731J

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