Benzoxaborole as a new chemotype for carbonic anhydrase inhibition-Reference-Cited by-同舟云学术

Benzoxaborole as a new chemotype for carbonic anhydrase inhibition

Published:2016 Issue:80 Volume:52 Page:11983-11986
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Alterio Vincenzo¹²³,Cadoni Roberta⁴⁵⁶⁷⁸,Esposito Davide¹²³,Vullo Daniela⁹¹⁰¹¹¹²¹³,Fiore Anna Di¹²³,Monti Simona Maria¹²³,Caporale Andrea¹²³^ORCID,Ruvo Menotti¹²³,Sechi Mario⁸¹⁴¹⁵³,Dumy Pascal⁴⁵⁶⁷,Supuran Claudiu T.¹⁶¹⁷¹¹¹³³,Simone Giuseppina De¹²³,Winum Jean-Yves⁴⁵⁶⁷

Affiliation:

1. Istituto di Biostrutture e Bioimagini-CNR

2. Naples

3. Italy

4. Institut des Biomolécules Max Mousseron (IBMM) UMR5247 CNRS, ENSCM

5. Université de Montpellier

6. Montpellier

7. France

8. Dipartimento di Chimica e Farmacia

9. Laboratorio di Chimica Bioinorganica

10. Polo Scientifico

11. Università degli Studi di Firenze

12. Sesto Fiorentino

13. Florence

14. Università degli Studi di Sassari

15. Sassari

16. Neurofarba Department

17. Section of Pharmaceutical and Nutriceutical Sciences

Abstract

In this paper we provide the first experimental evidence that benzoxaboroles can be used as CA inhibitors.

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2016/CC/C6CC06399C

Reference25 articles.

1. Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

2. Targeting Tumor Hypoxia: Suppression of Breast Tumor Growth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors

3. Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isoforms I and II and transmembrane, tumor-associated isoforms IX and XII with boronic acids

4. Carbonic anhydrase inhibitors. Inhibition of the fungal β-carbonic anhydrases from Candida albicans and Cryptococcus neoformans with boronic acids

5. 3D-QSAR-aided design, synthesis, in vitro and in vivo evaluation of dipeptidyl boronic acid proteasome inhibitors and mechanism studies

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