Synthesis of thiazolo[2,3-b]quinazoline derivatives via base-promoted cascade bicyclization of o-alkenylphenyl isothiocyanates with propargylamines-Reference-Cited by-同舟云学术

Synthesis of thiazolo[2,3-b]quinazoline derivatives via base-promoted cascade bicyclization of o-alkenylphenyl isothiocyanates with propargylamines

Published:2019 Issue:29 Volume:17 Page:6994-6997
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Miao Jiankang¹²³⁴⁵,Sang Xiaoyan¹²³⁴⁵,Wang Yi¹²³⁴⁵,Deng Shufeng¹²³⁴⁵,Hao Wenyan¹²³⁴⁵^ORCID

Affiliation:

1. Key Laboratory of Functional Small Organic Molecules

2. Ministry of Education

3. College of Chemistry & Chemical Engineering

4. Jiangxi Normal University

5. Nanchang

Abstract

A highly efficient base-promoted cascade bicyclization of o-alkenylphenyl isothiocyanates with propargylamines for constructing thiazolo[2,3-b]quinazolines has been demonstrated.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Jiangxi Province

Education Department of Jiangxi Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C9OB01098J

Reference50 articles.

1. Structure-Activity Relationship of Omeprazole and Analogs as Helicobacter pylori Urease Inhibitors

2. Discovery and Structure−Activity Relationship of the First Non-Peptide Competitive Human Glucagon Receptor Antagonists

3. Evaluation of 8-Arylsulfanyl, 8-Arylsulfoxyl, and 8-Arylsulfonyl Adenine Derivatives as Inhibitors of the Heat Shock Protein 90

4. Imino-tetrahydro-benzothiazole Derivatives as p53 Inhibitors: Discovery of a Highly Potent in Vivo Inhibitor and Its Action Mechanism

5. Synthesis, antitrichinnellosis and antiprotozoal activity of some novel thieno[2,3-d]pyrimidin-4(3H)-ones containing benzimidazole ring

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