Regioselective C–H sulfenylation of N-sulfonyl protected 7-azaindoles promoted by TBAI: a rapid synthesis of 3-thio-7-azaindoles-Reference-Cited by-同舟云学术

Regioselective C–H sulfenylation of N-sulfonyl protected 7-azaindoles promoted by TBAI: a rapid synthesis of 3-thio-7-azaindoles

Published:2020 Issue:53 Volume:10 Page:31819-31823
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Hu Jingyan¹²³⁴⁵,Ji Xiaoming¹²³⁴⁵,Hao Shuai¹²³⁴⁵,Zhao Mingqin¹²³⁴⁵,Lai Miao¹²³⁴⁵,Ren Tianbao¹²³⁴⁵,Xi Gaolei⁶⁷⁴⁵,Wang Erbin⁶⁷⁴⁵,Wang Juanjuan⁶⁷⁴⁵,Wu Zhiyong¹²³⁴⁵^ORCID

Affiliation:

1. Flavors and Fragrance Engineering & Technology Research Center of Henan Province

2. College of Tobacco Science

3. Henan Agricultural University

4. Zhengzhou

5. China

6. Technology Center

7. China Tobacco Henan Industrial Co., Ltd.

Abstract

A novel, practical and highly regioselective TBAI promoted C-3 sulfenylation reaction of N-sulfonyl protected 7-azaindoles with sulfonyl chlorides is presented here.

Funder

Henan Agricultural University

Education Department of Henan Province

Science and Technology Department of Henan Province

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/RA/D0RA06635D

Reference63 articles.

1. A New Family of Tunable Indolylphosphine Ligands by One-Pot Assembly and Their Applications in Suzuki−Miyaura Coupling of Aryl Chlorides