Progress in the development of small molecules as new human A3 adenosine receptor ligands based on the 3-thiophenylcoumarin core-Reference-Cited by-同舟云学术

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Progress in the development of small molecules as new human A3 adenosine receptor ligands based on the 3-thiophenylcoumarin core

Published:2016 Issue:5 Volume:7 Page:845-852
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Matos M. J.¹²³⁴⁵,Vilar S.⁶⁷⁸⁹¹⁰,Kachler S.¹¹¹²¹³¹⁴,Vazquez-Rodriguez S.¹²³⁴⁵,Varela C.¹⁵¹⁶⁷¹⁷⁵,Delogu G.¹⁸¹⁹²⁰²¹²²,Hripcsak G.²³²⁴²⁵²⁶,Santana L.⁶⁷⁸⁹¹⁰,Uriarte E.⁶⁷⁸⁹¹⁰,Klotz K.-N.¹¹¹²¹³¹⁴,Borges F.¹²³⁴⁵

Affiliation:

1. CIQUP/Department of Chemistry and Biochemistry

2. Faculty of Sciences

3. University of Porto

4. 4169-007 Porto

5. Portugal

6. Department of Organic Chemistry

7. Faculty of Pharmacy

8. University of Santiago de Compostela

9. 15782 Santiago de Compostela

10. Spain

11. Institute of Pharmacology and Toxicology

12. University of Würzburg

13. 97078 Würzburg

14. Germany

15. CNC-IBILI

16. Pharmaceutical Chemistry Group

17. University of Coimbra

18. Department of Life Sciences and Environment

19. Section of Pharmaceutical Sciences

20. University of Cagliari

21. 09124 Cagliari

22. Italy

23. Department of Biomedical Informatics

24. Columbia University Medical Center

25. New York

26. USA

Abstract

3-Thiophenylcoumarins are described as adenosine receptor ligands. Synthesis, in vitro pharmacological assays and docking studies were performed.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/MD/C5MD00573F

Reference29 articles.

1. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update

2. Mechanisms of induction of adenosine receptor genes and its functional significance

3. Adenosine Receptor Antagonists: Translating Medicinal Chemistry and Pharmacology into Clinical Utility

4. Adenosine and inflammation: what's new on the horizon?

5. Adenosine receptors: therapeutic aspects for inflammatory and immune diseases

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1. Cytogenotoxicity assessment of 3‐(3,4‐dihydroxyphenyl)‐7,8‐dihydroxycoumarin on HepG2/C3A cells and leukocytes;Journal of Applied Toxicology;2022-09-02

2. Adenosine Receptor Ligands: Coumarin–Chalcone Hybrids as Modulating Agents on the Activity of hARs;Molecules;2020-09-19

3. Descubrimiento de fármacos basado en imagenología de células vivas;Revista Colombiana de Ciencias Químico-Farmacéuticas;2020-01-01

4. Coumarins as Promising Scaffold for the Treatment of Age-related Diseases – An Overview of the Last Five Years;Current Topics in Medicinal Chemistry;2018-01-25

5. Coumarins and adenosine receptors: New perceptions in structure-affinity relationships;Chemical Biology & Drug Design;2017-09-04

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