Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as selective 5-HT7 receptor antagonists and their psychotropic properties-Reference-Cited by-同舟云学术

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Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as selective 5-HT7 receptor antagonists and their psychotropic properties

Published:2015 Issue:7 Volume:6 Page:1272-1277
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Zajdel Paweł¹²³⁴,Canale Vittorio¹²³⁴,Partyka Anna⁵²³⁴,Marciniec Krzysztof⁶⁷⁸⁴,Kurczab Rafał¹⁹¹⁰¹¹⁴,Satała Grzegorz¹⁹¹⁰¹¹⁴,Siwek Agata¹²²³⁴,Jastrzębska-Więsek Magdalena⁵²³⁴,Wesołowska Anna⁵²³⁴,Kos Tomasz¹³⁹¹⁰¹¹⁴,Popik Piotr¹³⁹¹⁰¹¹⁴,Bojarski Andrzej J.¹⁹¹⁰¹¹⁴

Affiliation:

1. Department of Medicinal Chemistry

2. Jagiellonian University Medical College

3. 30-688 Krakow

4. Poland

5. Department of Clinical Pharmacy

6. Department of Organic Chemistry

7. Medical University of Silesia

8. 41-200 Sosnowiec

9. Institute of Pharmacology

10. Polish Academy of Sciences

11. 31-343 Kraków

12. Department of Pharmacobiology

13. Department of Behavioral Neuroscience and Drug Development

Abstract

A novel series of potent 5-HT₇ receptor antagonist and their antidepressant, anxiolytic and pro-cognitive properties is described.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/MD/C5MD00166H

Reference36 articles.

1. Functional, molecular and pharmacological advances in 5-HT receptor research

2. The serotonin 5-HT7 receptors: two decades of research

3. Genetic knockout and pharmacological blockade studies of the 5-HT7 receptor suggest therapeutic potential in depression

4. 5-HT7 Receptor Inhibition and Inactivation Induce Antidepressantlike Behavior and Sleep Pattern

5. Enhancement of the anti-immobility action of antidepressants by a selective 5-HT7 receptor antagonist in the forced swimming test in mice

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1. The 5-HT7 receptor system as a treatment target for mood and anxiety disorders: A systematic review;Journal of Psychopharmacology;2023-11-23

2. Antidepressant Drug Discovery and Development: Mechanism and Drug Design Based on Small Molecules;Advanced Therapeutics;2022-03-30

3. Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties;Molecules;2021-06-23

4. Sustainable Synthesis of a Potent and Selective 5-HT7 Receptor Antagonist Using a Mechanochemical Approach;The Journal of Organic Chemistry;2020-07-24

5. Structure-activity relationships of serotonin 5-HT7 receptors ligands: A review;European Journal of Medicinal Chemistry;2019-12

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