Catalytic enantioselective one-pot approach tocis- andtrans-2,3-diaryl substituted 1,5-benzothiazepines-Reference-Cited by-同舟云学术

Catalytic enantioselective one-pot approach tocis- andtrans-2,3-diaryl substituted 1,5-benzothiazepines

Published:2018 Issue:38 Volume:16 Page:6923-6934
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Meninno Sara¹²³⁴^ORCID,Quaratesi Ilaria¹²³⁴,Volpe Chiara¹²³⁴,Mazzanti Andrea⁵⁶⁷⁴^ORCID,Lattanzi Alessandra¹²³⁴^ORCID

Affiliation:

1. Dipartimento di Chimica e Biologia “A. Zambelli”

2. Università di Salerno

3. Fisciano

4. Italy

5. Dipartimento di Chimica Industriale “Toso Montanari”

6. Università di Bologna

7. I-40136 Bologna

Abstract

A first enantioselective one-pot organocatalytic sulfa-Michael/lactamization sequence providedcis- andtrans-2,3-diaryl substituted 1,5-benzothiazepines in satisfactory yields and good to high enantioselectivity.

Funder

Università degli Studi di Salerno

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/OB/C8OB01988F

Reference45 articles.

1. 1,5-Benzothiazepine, a versatile pharmacophore: A review

2. Catalytic Approaches to Optically Active 1,5-Benzothiazepines

3. Benzothiazepines: chemistry of a privileged scaffold

4. Synthesis of optically active 1,5-benzothiazepines

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