1. For a recent discussion of transition state analogue design, see: P. R.Andrews and D. A.Winkler in ‘Drug Design: Fact or Fantasy,’ eds. G. Jolles and K. R. H. Wooldridge, Academic Press, New York, 1984, ch. 8.
2. Phosphonamidates as transition-state analog inhibitors of thermolysin
3. Evaluation of Intrinsic Binding Energy from a Hydrogen Bonding Group in an Enzyme Inhibitor
4. A. Meister in ‘The Enzymes,’ 3rd edn., vol. 10, ed. P. D. Boyer, Academic Press, 1974, New York, p. 699;