Synthesis of phosphaisocoumarin amidates via DIBAL-H-mediated selective amidation of phosphaisocoumarin esters-Reference-Cited by-同舟云学术

Synthesis of phosphaisocoumarin amidates via DIBAL-H-mediated selective amidation of phosphaisocoumarin esters

Published:2014 Issue:29 Volume:12 Page:5458-5463
ISSN:1477-0520
Container-title:Org. Biomol. Chem.
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Guo Yu-Juan¹²³,Chen Pei-Jiang¹²³,Wang Bo¹²³,Peng Ai-Yun¹²³

Affiliation:

1. School of Chemistry & Chemical Engineering

2. Sun Yat-sen University

3. Guangzhou, China

Abstract

A series of phosphaisocoumarin amidates were synthesized via DIBAL-H-mediated selective amidation of phosphaisocoumarin esters in good to excellent yields. In each case, the phostone ring was intact and only the exocyclic ethoxy group was amidated.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/OB/C4OB00663A

Reference35 articles.

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