Pd-Catalyzed highly selective and direct ortho C–H arylation of pyrrolo[2,3-d]pyrimidine derivatives-Reference-Cited by-同舟云学术

Pd-Catalyzed highly selective and direct ortho C–H arylation of pyrrolo[2,3-d]pyrimidine derivatives

Published:2020 Issue:2 Volume:7 Page:324-328
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Zhou Jing¹²³⁴,Mao Zhengtong¹²³⁴,Pan Haokun¹²³⁴,Zhang Xingxian¹²³⁴^ORCID

Affiliation:

1. College of Pharmaceutical Science

2. Zhejiang University of Technology

3. Hangzhou 310014

4. P. R. China

Abstract

Pd-Catalyzed one-pot direct ortho C–H arylation of pyrrolo[2,3-d]pyrimidine derivatives is reported. This protocol provides a variety of biphenyl-containing pyrrolo[2,3-d]pyrimidines in good to excellent yields.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/QO/C9QO01312A

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