One-pot mild and efficient synthesis of [1,3]thiazino[3,2-a]indol-4-ones and their anti-proliferative activity-Reference-Cited by-同舟云学术

One-pot mild and efficient synthesis of [1,3]thiazino[3,2-a]indol-4-ones and their anti-proliferative activity

Published:2019 Issue:16 Volume:17 Page:3914-3920
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Rhodes Steven¹²³⁴^ORCID,Short Spencer¹²³⁴^ORCID,Sharma Sidhika⁵⁶⁷⁸^ORCID,Kaur Ramneet⁵⁶⁷⁸^ORCID,Jha Mukund¹²³⁴^ORCID

Affiliation:

1. Department of Biology and Chemistry

2. Nipissing University

3. North Bay

4. Canada

5. Department of Biology

6. University of North Georgia

7. Oakwood

8. USA

Abstract

One-pot synthesis of [1,3]thiazino[3,2-a]indol-4-one frameworks is developed in aqueous medium and the anti-proliferative activity of the synthesized compounds is evaluated against two triple negative breast cancer cell lines.

Funder

Natural Sciences and Engineering Research Council of Canada

Nipissing University

Canada Foundation for Innovation

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C9OB00500E

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