Proteasome inhibition and cytostatic effects on human cancer cells by pyrazolone-enamines: a combined crystallographic, structural and computational study-Reference-Cited by-同舟云学术

Proteasome inhibition and cytostatic effects on human cancer cells by pyrazolone-enamines: a combined crystallographic, structural and computational study

Published:2015 Issue:3 Volume:39 Page:2168-2180
ISSN:1144-0546
Container-title:New Journal of Chemistry
language:en
Short-container-title:New J. Chem.

Author:

Yan Xingchen¹²³⁴⁵^ORCID,Xu Jiakun¹²³⁴⁵,Wu Xiaojing¹²³⁴⁵,Zhang Zhongyu¹²³⁴⁵,Zhang Xia¹²³⁴⁵,Fan Yuhua¹²³⁴⁵,Bi Caifeng¹²³⁴⁵

Affiliation:

1. Key Laboratory of Marine Chemistry Theory and Technology

2. Ministry of Education

3. College of Chemistry and Chemical Engineering

4. Ocean University of China

5. Qingdao

Abstract

Interactions are possibly through hydrogen bonding of the pyrazolone ring and the hydroxyl, or the intercalation of conjugated plane.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,General Chemistry,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2015/NJ/C4NJ01906G

Reference60 articles.

1. Synthesis, structural activity relationship and anti-tubercular activity of novel pyrazoline derivatives

2. Synthesis and antimycotic activity of N-azolyl-2,4-dihydroxythiobenzamides

3. Synthesis and investigation of anti-inflammatory activity and gastric ulcerogenicity of novel nitric oxide-donating pyrazoline derivatives

4. Identification of antibacterial and antifungal pharmacophore sites for potent bacteria and fungi inhibition: Indolenyl sulfonamide derivatives

5. Development of selective and reversible pyrazoline based MAO-B inhibitors: Virtual screening, synthesis and biological evaluation

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