“Seasoning” antimalarial drugs' action: chloroquine bile salts as novel triple-stage antiplasmodial hits

Author:

Silva Ana Teresa1,Oliveira Isabel2,Duarte Denise3ORCID,Moita Diana4,Prudêncio Miguel4ORCID,Nogueira Fátima3,Ferraz Ricardo15ORCID,Marques Eduardo Figueira2ORCID,Gomes Paula1ORCID

Affiliation:

1. LAQV-REQUIMTE, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, P-4169-007 Porto, Portugal

2. CIQUP - IMS, Departamento de Química e Bioquímica, Faculdade de Ciências, Universidade do Porto, P-4169-007 Porto, Portugal

3. Global Health and Tropical Medicine, Instituto de Higiene e Medicina Tropical, Universidade Nova de Lisboa, P-1349-008 Lisboa, Portugal

4. Instituto de Medicina Molecular, Faculdade de Medicina Universidade de Lisboa, P-1649 028 Lisboa, Portugal

5. Ciências Químicas e das Biomoléculas, Escola Superior de Saúde - Instituto Politécnico do Porto, P-4200-072 Porto, Portugal

Abstract

Malaria is one of the “big three” global infectious diseases, with the heaviest toll on human lives in low-to-middle income countries. Cost-effective antimalarial drugs with multi-stage action remain an unmet and urgent need in global healthcare.

Funder

Fundação para a Ciência e a Tecnologia

Publisher

Royal Society of Chemistry (RSC)

Reference40 articles.

1. “Big Three” Infectious Diseases: Tuberculosis, Malaria and HIV/AIDS

2. https://www.un.org/sustainabledevelopment/health/ (assessed on Dec. 29th 2023 )

3. World Health Organization , World Malaria Report 2021 , World Health Organization , Geneva , 2021

4. World Health Organization , Malaria eradication: benefits, future scenarios, and feasibility: a report of the Strategic Advisory Group on Malaria Eradication , 2020

5. Has artemisinin resistance emerged in Africa?

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