Stereoselective synthesis of trans-aziridines via intramolecular oxidative C(sp3)–H amination of β-amino ketones-Reference-Cited by-同舟云学术

Stereoselective synthesis of trans-aziridines via intramolecular oxidative C(sp3)–H amination of β-amino ketones

Published:2020 Issue:5 Volume:7 Page:780-786
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Tan Chen¹²³⁴⁵,Liu Yongguo⁶⁷⁸⁵,Liu Xinyuan¹²³⁴⁵,Jia Huanxin¹²³⁴⁵,Xu Kun⁹¹⁰¹¹⁵^ORCID,Huang Sihan¹²³⁴⁵,Wang Jingwen¹²³⁴⁵,Tan Jiajing¹²³⁴⁵^ORCID

Affiliation:

1. Department of Organic Chemistry

2. College of Chemistry

3. Beijing University of Chemical Technology

4. Beijing 100029

5. China

6. Beijing Key Laboratory of Flavor Chemistry

7. Beijing Technology and Business University (BTBU)

8. Beijing 100048

9. College of Chemistry and Pharmaceutical Engineering

10. Nanyang Normal University

11. Nanyang

Abstract

An expedient strategy for the synthesis of trans-2,3-disubstituted via the intramolecular KI/TBHP mediated oxidative dehydrogenative C(sp³)–H amination reaction was presented.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Beijing Municipality

Fundamental Research Funds for the Central Universities

Beijing Technology and Business University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/QO/C9QO01489F

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