Efficient Pd-catalyzed domino synthesis of 1-phenyl-1H-indol-2-amine and 5-amino-indolo[1,2-a]quinazoline derivatives-Reference-Cited by-同舟云学术

Efficient Pd-catalyzed domino synthesis of 1-phenyl-1H-indol-2-amine and 5-amino-indolo[1,2-a]quinazoline derivatives

Published:2015 Issue:40 Volume:13 Page:10122-10126
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Jiang Min¹²³⁴⁵,Xiang Haoyue⁶⁷⁸⁵⁹,Zhu Fangxia¹²³⁴⁵,Xu Xing¹²³⁴⁵,Deng Lianfu¹²³⁴⁵,Yang Chunhao⁶⁷⁸⁵⁹

Affiliation:

1. Shanghai Key Laboratory for Bone and Joint Diseases

2. Shanghai Institute of Traumatology and Orthopaedics

3. Shanghai Ruijin Hospital

4. Shanghai Jiaotong University School of Medicine

5. Shanghai

6. State Key Laboratory of Drug Research

7. Shanghai Institute of Materia Medica

8. Chinese Academy of Sciences

9. P. R. China

Abstract

Efficient and practical access to 1-phenyl-1H-indol-2-amine and 5-amino-indolo[1,2-a]quinazoline derivatives is presented via a Buchwald–Hartwig type coupling and a base-promoted intramolecular nucleophilic reaction.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB01642H

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5. Discovery of a Potent and Selective Protein Kinase CK2 Inhibitor by High-Throughput Docking

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