Catalytic asymmetric Michael/cyclization reaction of 3-isothiocyanato thiobutyrolactone: an approach to the construction of a library of bispiro[pyrazolone-thiobutyrolactone] skeletons-Reference-Cited by-同舟云学术

Catalytic asymmetric Michael/cyclization reaction of 3-isothiocyanato thiobutyrolactone: an approach to the construction of a library of bispiro[pyrazolone-thiobutyrolactone] skeletons

Published:2022 Issue:25 Volume:20 Page:5060-5065
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Liu Ren-Ming¹,Zhang Min¹,Han Xiao-Xue¹,Liu Xiong-Li¹^ORCID,Pan Bo-Wen²,Tian You-Ping²,Peng Li-Jun¹,Yuan Wei-Cheng³^ORCID

Affiliation:

1. National & Local Joint Engineering Research Center for the Exploitation of Homology Resources of Southwest Medicine and Food, Guizhou University, Guiyang, Guizhou 550025, P. R. China

2. College of Pharmaceutical Sciences, Guizhou University of Traditional Chinese Medicine, Guiyang, 550025, China

3. Innovation Research Center of Chiral Drugs, Institute for Advanced Study, School of Pharmacy, Chengdu University, Chengdu 610106, China

Abstract

Here, we demonstrate the first example of 3-isothiocyanato thiobutyrolactone serving as a useful building block in the Michael/cyclization reaction.

Funder

Data Center of Management Science, National Natural Science Foundation of China - Peking University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/OB/D2OB00773H

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