Synthesis and binding affinities for sst receptors of cyclic peptoid SRIF-mimetics-Reference-Cited by-同舟云学术

Synthesis and binding affinities for sst receptors of cyclic peptoid SRIF-mimetics

Published:2012 Issue:12 Volume:3 Page:1531-1535
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Caumes Cécile¹²³⁴⁵,Hjelmgaard Thomas¹²³⁴⁵,Roy Olivier¹²³⁴⁵,Reynaud Morgane⁶⁷⁸⁹⁵,Servent Denis⁶⁷⁸⁹⁵,Taillefumier Claude¹²³⁴⁵,Faure Sophie¹²³⁴⁵

Affiliation:

1. Clermont Universités

2. Université Blaise Pascal

3. Institut de Chimie de Clermont-Ferrand (ICCF)

4. 63000 Clermont-Ferrand

5. France

6. CEA

7. iBiTecS

8. Service d'Ingénierie Moléculaire des Protéines (SIMOPRO)

9. 91191 Gif sur Yvette

Abstract

Synthesis of the first all-peptoid SRIF (Somatotropin Release-Inhibiting Factor) analogues and evaluation of their binding affinities for the five human somatostatin receptors (hsst1–5).

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2012/MD/C2MD20265D

Reference65 articles.

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2. Opportunities in somatostatin research: biological, chemical and therapeutic aspects

3. Cloning and functional characterization of a family of human and mouse somatostatin receptors expressed in brain, gastrointestinal tract, and kidney.

4. In Vivo and in Vitro Plasma Disappearance and Metabolism of Somatostatin-28 and Somatostatin-14 in the Rat*

5. Biologic and immunologic activities and applications of somatostatin analogs

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