Pd(ii)-catalyzed, controllable C–H mono-/diarylation of aryl tetrazoles: concise synthesis of Losartan
Author:
Affiliation:
1. Department of Chemistry
2. University of Science and Technology of China
3. Hefei
4. China
Abstract
A palladium(ii)-catalyzed C–H arylation directed by tetrazole has been developed with excellent mono-/di-selectivity through adjustment of the protecting site on the tetrazole ring.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/OB/C4OB02453B
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