Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H3 receptor antagonists-Reference-Cited by-同舟云学术

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Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H3 receptor antagonists

Published:2019 Issue:2 Volume:10 Page:234-251
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Staszewski Marek¹²³⁴^ORCID,Stasiak Anna⁵²⁶⁴,Karcz Tadeusz⁷⁸⁹¹⁰⁴,McNaught Flores Daniel¹¹¹²¹³¹⁴¹⁵,Fogel Wiesława Agnieszka⁵²⁶⁴^ORCID,Kieć-Kononowicz Katarzyna⁷⁸⁹¹⁰⁴^ORCID,Leurs Rob¹¹¹²¹³¹⁴¹⁵,Walczyński Krzysztof¹²³⁴^ORCID

Affiliation:

1. Department of Synthesis and Technology of Drugs

2. Medical University of Lodz

3. 90-151 Łódź

4. Poland

5. Department of Hormone Biochemistry

6. 90-752 Łódź

7. Department of Technology and Biotechnology of Drugs

8. Faculty of Pharmacy

9. Jagiellonian UniversityMedical College

10. 30-688 Kraków

11. Amsterdam Institute of Molecules

12. Medicines & Systems, Division of Medicinal Chemistry

13. Vrije Universiteit Amsterdam

14. 1081 HZ Amsterdam

15. The Netherlands

Abstract

The prominent members of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines as histamine H₃ receptor antagonists.

Funder

Uniwersytet Medyczny w Lodzi

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/MD/C8MD00527C

Reference44 articles.

1. Genomics Meets Histamine Receptors: New Subtypes, New Receptors

2. The role of histamine H4 receptor in immune and inflammatory disorders

3. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

4. H3-Receptors Control Histamine Release in Human Brain

5. Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats

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1. 3D-QSAR and Pharmacophoric study on 2,6-Disubstituted Thiazolo [4,5-b] Pyridines as H3 Receptor Antagonists;Research Journal of Pharmacy and Technology;2023-10-31

2. Dual Targeting Ligands—Histamine H3 Receptor Ligands with Monoamine Oxidase B Inhibitory Activity—In Vitro and In Vivo Evaluation;Pharmaceutics;2022-10-13

3. Guanidine Derivatives: How Simple Structural Modification of Histamine H3R Antagonists Has Led to the Discovery of Potent Muscarinic M2R/M4R Antagonists;ACS Chemical Neuroscience;2021-06-08

4. Synthesis, structure and catalytic activity of rare-earth metal amino complexes incorporating imino-functionalized indolyl ligand;Journal of Organometallic Chemistry;2021-02

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