Straightforward synthesis of N-arylindoles via one-pot Fischer indolisation–indole N-arylation-Reference-Cited by-同舟云学术

Straightforward synthesis of N-arylindoles via one-pot Fischer indolisation–indole N-arylation

Published:2023 Issue:23 Volume:13 Page:15993-15997
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Lintott Mia¹,Perry Alexis¹^ORCID

Affiliation:

1. Biosciences, University of Exeter, Stocker Road, Exeter EX4 4QD, UK

Abstract

One-pot, microwave-promoted Fischer indolisation–indole N-arylation enables straightforward, rapid synthesis of structurally-diverse N-arylindoles from widely-available precursors, using a simple, air-stable catalyst in a common, sustainable solvent.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2023/RA/D3RA02658B

Reference56 articles.

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5. Unprecedented Stereocontrol in the Synthesis of 1,2,3-Trisubstituted Tetrahydro-β-carbolines through an Asymmetric Pictet-Spengler Reaction towards Sarpagine-Type Indole Alkaloids

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