InCl3-catalyzed 5-exo-dig cyclization/1,6-conjugate addition of N-propargylamides with p-QMs to construct oxazole derivatives-Reference-Cited by-同舟云学术

InCl3-catalyzed 5-exo-dig cyclization/1,6-conjugate addition of N-propargylamides with p-QMs to construct oxazole derivatives

Published:2020 Issue:9 Volume:18 Page:1780-1784
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Nan Guang-Ming¹²³⁴,Li Xue¹²³⁴,Yao Tian-Yu⁵⁶⁷⁸⁴,Yan Ting-Xun⁵⁶⁷⁸⁴,Wen Li-Rong⁵⁶⁷⁸⁴^ORCID,Li Ming¹²³⁴⁵^ORCID

Affiliation:

1. University and College Key Lab of Natural Product Chemistry and Application in Xinjiang

2. Yili Normal University

3. Yining 835000

4. China

5. State Key Laboratory Base of Eco-Chemical Engineering

6. College of Chemistry and Molecular Engineering

7. Qingdao University of Science & Technology

8. Qingdao 266042

Abstract

An InCl₃-catalyzed tandem intramolecular 5-exo-dig cyclization/1,6-conjugate addition/aromatization of N-propargylamides with p-QMs to produce oxazoles tethering diarylmethane has been successfully developed.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Shandong Province

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/OB/C9OB02651G

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5. Muscarine, imidazole, oxazole and thiazole alkaloids

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