Iridium-catalysed C–H borylation of β-aryl-aminopropionic acids-Reference-Cited by-同舟云学术

Iridium-catalysed C–H borylation of β-aryl-aminopropionic acids

Published:2020 Issue:34 Volume:18 Page:6696-6701
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Robinson Henry¹²³⁴⁵,Stillibrand Joe¹²³⁴⁵,Simelis Klemensas¹²³⁴⁵,Macdonald Simon J. F.⁶⁷⁸⁵,Nortcliffe Andrew¹²³⁴⁵^ORCID

Affiliation:

1. GlaxoSmithKline Carbon Neutral Laboratories for Sustainable Chemistry

2. School of Chemistry

3. University of Nottingham

4. Nottingham

5. UK

6. GlaxoSmithKline

7. Medicines Research Centre

8. Stevenage

Abstract

Iridium-catalysed C–H borylation of β-aryl-aminopropionic acid derivatives gives 3,5-functionalised protected β-aryl-aminopropionic acid boronates. One-pot borylation–functionalisation provides diverse building blocks for medicinal chemistry.

Funder

University of Nottingham

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/OB/D0OB01495H

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