Rapid 18F-labeling via Pd-catalyzed S-arylation in aqueous medium-Reference-Cited by-同舟云学术

Rapid 18F-labeling via Pd-catalyzed S-arylation in aqueous medium

Published:2021 Issue:29 Volume:57 Page:3547-3550
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Humpert Swen¹²³⁴⁵^ORCID,Omrane Mohamed A.¹²³⁴⁵,Urusova Elizaveta A.¹²³⁴⁵,Gremer Lothar⁶⁷⁸⁹⁵^ORCID,Willbold Dieter⁶⁷⁸⁹⁵^ORCID,Endepols Heike¹²³⁴⁵^ORCID,Krasikova Raisa N.¹⁰¹¹¹²¹³¹⁴^ORCID,Neumaier Bernd¹²³⁴⁵^ORCID,Zlatopolskiy Boris D.¹²³⁴⁵^ORCID

Affiliation:

1. Institute of Neuroscience and Medicine

2. Nuclear Chemistry (INM-5)

3. Forschungszentrum Jülich GmbH

4. Jülich 52428

5. Germany

6. Institute of Biological Information Processing

7. Structural Biochemistry (IBI-7)

8. Forschungszentrum Jülich

9. Jülich 52425

10. N. P. Bechtereva Institute of the Human Brain

11. St.-Petersburg 197376

12. Russia

13. St.-Petersburg State University

14. St.-Petersburg 199034

Abstract

Rapid Pd-catalyzed S-arylation with easily accessible 2-[¹⁸F]fluoro-5-iodopyridine enables facile preparation of radiolabeled peptides and proteins.

Funder

Russian Foundation for Basic Research

Deutsche Forschungsgemeinschaft

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2021/CC/D1CC00745A

Reference35 articles.

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