Demonstration of the dynamic mass redistribution label-free technology as a useful cell-based pharmacological assay for endogenously expressed GABAA receptors-Reference-Cited by-同舟云学术

Demonstration of the dynamic mass redistribution label-free technology as a useful cell-based pharmacological assay for endogenously expressed GABAA receptors

Published:2016 Issue:3 Volume:7 Page:426-432
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Klein Anders B.¹²³⁴⁵,Nittegaard-Nielsen Mia¹²³⁴⁵,Christensen Julie T.¹²³⁴⁵,Al-Khawaja Anas¹²³⁴⁵,Wellendorph Petrine¹²³⁴⁵^ORCID

Affiliation:

1. Department of Drug Design and Pharmacology

2. Faculty of Health and Medical Sciences

3. University of Copenhagen

4. DK-2100 Copenhagen

5. Denmark

Abstract

Within the continuous quest for the discovery of pharmacologically interesting compounds, the development of new and superior drug screening assays is desired.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/MD/C5MD00442J

Reference24 articles.

1. Variations on an inhibitory theme: phasic and tonic activation of GABAA receptors

2. Enhancement of GABAergic Activity: Neuropharmacological Effects of Benzodiazepines and Therapeutic Use in Anesthesiology

3. Beyond classical benzodiazepines: novel therapeutic potential of GABAA receptor subtypes

4. Structure, Function, and Modulation of GABAA Receptors

5. Comparing Label-Free Biosensors for Pharmacological Screening With Cell-Based Functional Assays

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