Construction of benzofuranone library via a metal-free, one-pot intermolecular condensation, and their application as efficient estrogen receptor β modulators-Reference-Cited by-同舟云学术

Construction of benzofuranone library via a metal-free, one-pot intermolecular condensation, and their application as efficient estrogen receptor β modulators

Published:2019 Issue:97 Volume:55 Page:14570-14573
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Peng Xueke¹²³⁴⁵,Hu Zhiye¹²³⁴⁵,Zhang Jing¹²³⁴⁵,Ning Wentao¹²³⁴⁵,Zhang Silong¹²³⁴⁵,Dong Chune¹²³⁴⁵^ORCID,Shi Xiaodong⁶⁷⁸⁹^ORCID,Zhou Hai-Bing¹²³⁴⁵^ORCID

Affiliation:

1. State Key Laboratory of Virology

2. Key Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University)

3. Ministry of Education

4. Hubei Province Engineering and Technology Research Center for Fluorinated Pharmaceuticals

5. Wuhan University School of Pharmaceutical Sciences

6. Department of Chemistry

7. University of South Florida

8. Tampa

9. USA

Abstract

Facile synthesis of benzofuranones as efficient estrogen receptor β modulators was achieved through a metal-free, one-pot intermolecular condensation between α-hydroxy aryl ketones and resorcinol derivatives.

Funder

National Natural Science Foundation of China

Wuhan University

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2019/CC/C9CC05756K

Reference29 articles.

1. Estrogen Receptors: How Do They Signal and What Are Their Targets

2. What pharmacologists can learn from recent advances in estrogen signalling

3. Cloning of the human estrogen receptor cDNA.

4. Cloning of a novel receptor expressed in rat prostate and ovary.

5. Predictive features of ligand‐specific signaling through the estrogen receptor

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