Design, synthesis and biological evaluation of imidazopyridine–propenone conjugates as potent tubulin inhibitors-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of imidazopyridine–propenone conjugates as potent tubulin inhibitors

Published:2017 Issue:5 Volume:8 Page:1000-1006
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Sayeed Ibrahim Bin¹²³⁴⁵,Lakshma Nayak V.¹²³⁴,Shareef Mohd Adil¹²³⁴,Chouhan Neeraj Kumar¹²³⁴,Kamal Ahmed¹²³⁴^ORCID

Affiliation:

1. Medicinal Chemistry and Pharmacology Division

2. CSIR - Indian Institute of Chemical Technology

3. Hyderabad 500007

4. India

5. Academy of Scientific and Innovative Research (AcSIR)

Abstract

A library of imidazopyridine–propenone conjugates (8a–8u) were synthesized and evaluated for their antitumor activity against four human cancer cell lines.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/MD/C7MD00043J

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