Diaminodiacid-based synthesis of macrocyclic peptides using 1,2,3-triazole bridges as disulfide bond mimetics-Reference-Cited by-同舟云学术

Diaminodiacid-based synthesis of macrocyclic peptides using 1,2,3-triazole bridges as disulfide bond mimetics

Published:2017 Issue:4 Volume:7 Page:2110-2114
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Guo Ye¹²³⁴⁵,Liu Chao¹²³⁴⁵,Song Hui²⁶⁷⁵,Wang Feng-Liang⁸⁹¹⁰⁵,Zou Yan¹²³⁴⁵,Wu Qiu-Ye¹²³⁴⁵,Hu Hong-Gang¹²³⁴⁵^ORCID

Affiliation:

1. Department of Organic Chemistry

2. College of Pharmacy

3. Second Military Medical University

4. Shanghai 200433

5. China

6. Weifang Medical University

7. Weifang

8. Department of Pharmacy

9. Baotou Medical College

10. Baotou

Abstract

A new approach for the efficient construction of 1,2,3-triazole bridges as disulfide surrogates in peptides, utilizing the diaminodiacid strategy was established.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/RA/C6RA26617G

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