Chloroquinoline–acetamide hybrids: a promising series of potential antiprotozoal agents-Reference-Cited by-同舟云学术

Chloroquinoline–acetamide hybrids: a promising series of potential antiprotozoal agents

Published:2015 Issue:60 Volume:5 Page:48368-48381
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Inam Afreen¹²³⁴,Van Zyl Robyn L.⁵⁶⁷⁸⁹,van Vuuren Natasha J.⁵⁶⁷⁸⁹,Chen Chien-Teng⁵⁶⁷⁸⁹,Avecilla Fernando¹⁰¹¹¹²¹³¹⁴,Agarwal Subhash M.¹⁵¹⁶¹⁷⁴,Azam Amir¹²³⁴

Affiliation:

1. Department of Chemistry

2. Jamia Millia Islamia

3. New Delhi

4. India

5. Pharmacology Division

6. Department of Pharmacy and Pharmacology

7. WITS Research Institute for Malaria (WRIM)

8. Faculty of Health Sciences

9. University of Witwatersrand

10. Departamento de Química Fundamental

11. Universidade da Coruña

12. Campus da Zapateira

13. 15071 A Coruña

14. Spain

15. Bioinformatics Division

16. Institute of Cytology and Preventive Oncology (ICMR) I-7

17. Noida 201301

Abstract

In an endeavour to develop efficacious antiprotozoal agents chloroquinoline–acetamide hybrids were synthesized and screened in vitro against E. histolytica and P. falciparum and molecular docking studies were performed against PfDHFR.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/RA/C5RA05472A

Reference60 articles.

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