Synthesis of amino heterocycle aspartyl protease inhibitors
Author:
Affiliation:
1. The Walter and Eliza Hall Institute for Medical Research
2. Parkville
3. Australia
4. Merck Research Laboratories
5. Kenilworth
6. 07033 USA
7. West Point
8. USA
9. The University of Melbourne
Abstract
Synthetic strategies to access 2-amino heterocycle head groups that inhibit aspartyl proteases, are reviewed.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2016/OB/C5OB01842K
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