Transition-metal-free highly regioselective C–H acetoxylation of pyrrolo[2,3-d]pyrimidine derivatives-Reference-Cited by-同舟云学术

Transition-metal-free highly regioselective C–H acetoxylation of pyrrolo[2,3-d]pyrimidine derivatives

Published:2020 Issue:18 Volume:7 Page:2696-2702
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Mao Zhengtong¹²³⁴,Liu Min¹²³⁴,Zhu Gaoyang¹²³⁴,Zhou Jing¹²³⁴,Zhang Xingxian¹²³⁴^ORCID

Affiliation:

1. College of Pharmaceutical Science

2. Zhejiang University of Technology

3. Hangzhou 310014

4. P. R. China

Abstract

Transition-metal-free catalyzed direct C(sp²)–H acetoxylation of pyrrolo[2,3-d]pyrimidine derivatives is reported. This protocol provides a variety of acetoxylated pyrrolo[2,3-d]pyrimidines in good to excellent yields.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/QO/D0QO00702A

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