Design and synthesis of cenocladamide analogues and their evaluation against breast cancer cell lines
Author:
Affiliation:
1. Departamento de Química Orgânica Instituto de Química
2. Universidade Estadual de Campinas (Unicamp)
3. Campinas
4. Brazil
5. Laboratório Nacional de Biociências (LNBio)
6. Centro Nacional de Pesquisa em Energia e Materiais (CNPEM)
Abstract
Synthesis of a concise series based on the natural product cenocladamide, their evaluation against a panel of breast cancer cells and preliminary mechanistic studies are discussed in this work.
Funder
Fundo de Apoio ao Ensino, à Pesquisa e Extensão, Universidade Estadual de Campinas
Fundação de Amparo à Pesquisa do Estado de São Paulo
Conselho Nacional de Desenvolvimento Científico e Tecnológico
Publisher
Royal Society of Chemistry (RSC)
Subject
Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2017/MD/C6MD00577B
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