Curcumin-based pyrazoline analogues as selective inhibitors of human monoamine oxidase A-Reference-Cited by-同舟云学术

Curcumin-based pyrazoline analogues as selective inhibitors of human monoamine oxidase A

Published:2018 Issue:7 Volume:9 Page:1164-1171
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Nath Chandrani¹²³⁴,Badavath Vishnu Nayak¹²³⁴,Thakur Abhishek⁵⁶⁷⁸,Ucar Gulberk⁹¹⁰¹¹¹²¹³,Acevedo Orlando⁵⁶⁷⁸^ORCID,Mohd Siddique Mohd Usman¹²³⁴,Jayaprakash Venkatesan¹²³⁴^ORCID

Affiliation:

1. Department of Pharmaceutical Sciences & Technology

2. Birla Institute of Technology

3. Ranchi-835 215

4. India

5. Department of Chemistry

6. University of Miami

7. Coral Gables

8. USA

9. Department of Biochemistry

10. Faculty of Pharmacy

11. Hacettepe University

12. Ankara

13. Turkey

Abstract

Chlorine substitution on a 3,5-diphenyl-pyrazoline derivative enabled potent and selective inhibition of hMAO-A; calculations suggest an “aromatic sandwich” orientation is responsible.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2018/MD/C8MD00196K

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