Selective synthesis of 3-deoxy-5-hydroxy-1-amino-carbasugars as potential α-glucosidase inhibitors-Reference-Cited by-同舟云学术

Selective synthesis of 3-deoxy-5-hydroxy-1-amino-carbasugars as potential α-glucosidase inhibitors

Published:2019 Issue:21 Volume:17 Page:5381-5391
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Jiang Chunfeng¹²³⁴⁵,Liu Quan⁶⁷⁵,Liu Jiaming¹²³⁴⁵,Liu Kaixuan¹²³⁴⁵,Tian Liangliang¹²³⁴⁵,Duan Mingfei¹²³⁴⁵,Wang Ying¹²³⁴⁵,Shen Zhufang⁶⁷⁵^ORCID,Xu Youjun¹²³⁴⁵^ORCID

Affiliation:

1. School of Pharmaceutical Engineering

2. and Key Laboratory of Structure-Based Drug Design & Discovery (Ministry of Education)

3. Shenyang Pharmaceutical University

4. Shenyang 110016

5. P. R. China

6. Chinese Academy of Medical Sciences and Peking Union Medical College

7. Beijing 100050

Abstract

A selective synthesis of 13 and 15, which could be converted to carbasugars as α-glucosidase inhibitors, was developed.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C9OB00762H

Reference21 articles.

1. Alicyclic Carbohydrates. XXIX.1,2 The Synthesis of a Pseudo-Hexose (2,3,4,5-Tetrahydroxycyclohexanemethanol)

2. Selective glycosidase inhibitors: A patent review (2012–present)

3. Glycosidase inhibitors: a patent review (2008 – 2013)

4. Recent developments in design and synthesis of bicyclic azasugars, carbasugars and related molecules as glycosidase inhibitors

5. Synthesis and Conformational and Biological Aspects of Carbasugars

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