Copper-assisted synthesis of dihydropyrano[2.3-b]indole-4-ones by domino cascade reaction-Reference-Cited by-同舟云学术

Copper-assisted synthesis of dihydropyrano[2.3-b]indole-4-ones by domino cascade reaction

Published:2021 Issue:12 Volume:19 Page:2692-2702
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Luo Yang¹²³⁴⁵,Zhong Xue¹²³⁴⁵,Huang Jiang-Kun¹²³⁴⁵,He Ling¹²³⁴⁵^ORCID

Affiliation:

1. Key Laboratory of Drug-Targeting and Drug Delivery System of the Education Ministry

2. Sichuan Engineering Laboratory for Plant-Sourced Drug and Sichuan Research Center for Drug Precision Industrial Technology

3. Department of Medicinal Chemistry

4. West China School of Pharmacy

5. Sichuan University

Abstract

A novel copper-catalyzed cascade intermolecular and intramolecular oxidation/cyclization domino one-pot reaction process for the regioselective synthesis of dihydropyrano[2.3-b]indol-4(9H)-ones has been successfully developed.

Funder

National Natural Science Foundation of China

Sichuan University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/OB/D1OB00078K

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3. Resolution of etodolac and antiinflammatory and prostaglandin synthetase inhibiting properties of the enantiomers

4. Synthesis and analgesic activity of pemedolac [cis-1-ethyl-1,3,4,9-tetrahydro-4-(phenylmethyl)pyrano[3,4-b]indole-1-acetic acid]

5. Discovery of Pyrano[3,4-b]indoles as Potent and Selective HCV NS5B Polymerase Inhibitors

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