Investigation on the reactivity of nucleophilic radiohalogens with arylboronic acids in water: access to an efficient single-step method for the radioiodination and astatination of antibodies
Author:
Affiliation:
1. Université de Nantes
2. CNRS
3. Inserm
4. CRCINA
5. F-44000 Nantes
6. CRNH-O
7. Mass Spectrometry Core Facility
8. France
9. NUN
Abstract
The high reactivity of astatine and iodine in water with arylboronic acids provides access to an efficient single-step antibody radiolabelling.
Funder
Agence Nationale de la Recherche
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2021/SC/D0SC05191H
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