Catalyst- and solvent-free, pot, atom and step economic synthesis of tetrahydroquinazolines by an aza-Diels–Alder reaction strategy
Author:
Affiliation:
1. Medicinal Chemistry Division
2. CSIR-North-East Institute of Science & Technology
3. Jorhat, India
4. Department of Chemistry
5. Nalbari College
6. Nalbari, India
Abstract
2,4-Disubstituted tetrahydroquinazolines can be readily obtained via a four-component aza-Diels–Alder reaction inside a microwave reactor. The methodology developed is simple, catalyst- and solvent-free and can be tuned to get dihydroquinazoline derivatives.
Publisher
Royal Society of Chemistry (RSC)
Subject
Pollution,Environmental Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2014/GC/C3GC42389A
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