Efficient microwave-assisted Suzuki–Miyaura cross-coupling reaction of 3-bromo pyrazolo[1,5-a]pyrimidin-5(4H)-one: towards a new access to 3,5-diarylated 7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine derivatives-Reference-Cited by-同舟云学术

Efficient microwave-assisted Suzuki–Miyaura cross-coupling reaction of 3-bromo pyrazolo[1,5-a]pyrimidin-5(4H)-one: towards a new access to 3,5-diarylated 7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine derivatives

Published:2021 Issue:3 Volume:11 Page:1287-1302
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Jismy Badr¹²³⁴,Guillaumet Gérald⁵⁶⁷⁴,Akssira Mohamed⁸⁹¹⁰¹¹,Tikad Abdellatif¹²²¹³¹⁴¹⁵,Abarbri Mohamed¹²³⁴^ORCID

Affiliation:

1. Laboratoire de Physico-Chimie des Matériaux et des Electrolytes pour l'Energie (PCM2E). EA 6299

2. Faculté des Sciences

3. 37200 Tours

4. France

5. Institut de Chimie Organique et Analytique (ICOA)

6. Université d'Orléans

7. UMR CNRS 7311

8. Laboratoire de Chimie Physique et de Chimie Bioorganique

9. URAC 22

10. 28800 Mohammedia

11. Morocco

12. Laboratoire de Chimie Moléculaire et Substances Naturelles

13. Département de Chimie

14. Université Moulay Ismail

15. Meknès 50050

Abstract

A convenient and efficient synthetic route to C3-arylated 7-trifluoromethylpyrazolo[1,5-a]pyrimidin-5-one derivatives has been reported starting from 3-bromo-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-one through a Suzuki–Miyaura cross-coupling reaction.

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/RA/D0RA07959F

Reference123 articles.

1. Palladium-Catalyzed Cross-Coupling: A Historical Contextual Perspective to the 2010 Nobel Prize

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