Copper-catalyzed asymmetric 1,2-arylboration of enamines: access to chiral borate-containing 3,3′-disubstituted isoindolinones-Reference-Cited by-同舟云学术

Copper-catalyzed asymmetric 1,2-arylboration of enamines: access to chiral borate-containing 3,3′-disubstituted isoindolinones

Published:2024 Issue:30 Volume:22 Page:6085-6089
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Xie Jia-Qi¹,Wang Bing-Xia¹,Liang Ren-Xiao¹^ORCID,Jia Yi-Xia¹²^ORCID

Affiliation:

1. College of Chemical Engineering, State Key Laboratory Breeding Base of Green-Chemical Synthesis Technology, Zhejiang University of Technology, Chaowang Road 18#, Hangzhou 310014, China

2. School of Chemistry and Chemical Engineering, Tianjin University of Technology, Tianjin 300384, China

Abstract

An enantioselective Cu-catalyzed 1,2-arylboration reaction of N-(o-iodobenzoyl)enamines with bis(pinacolato)diboron (B2pin2) is developed to access chiral borate-containing 3,3′-disubstituted isoindolinones.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Zhejiang Province

Fundamental Research Funds for the Provincial Universities of Zhejiang

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/OB/D4OB00896K

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