Microwave-assisted preparation of 4-amino-3-cyano-5-methoxycarbonyl-N-arylpyrazoles as building blocks for the diversity-oriented synthesis of pyrazole-based polycyclic scaffolds-Reference-Cited by-同舟云学术

Microwave-assisted preparation of 4-amino-3-cyano-5-methoxycarbonyl-N-arylpyrazoles as building blocks for the diversity-oriented synthesis of pyrazole-based polycyclic scaffolds

Published:2015 Issue:2 Volume:13 Page:409-423
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Corre Laurent Le¹²³⁴⁵,Tak-Tak Lotfi¹²³⁴⁵,Guillard Arthur¹²³⁴⁵,Prestat Guillaume¹²³⁴⁵,Gravier-Pelletier Christine¹²³⁴⁵,Busca Patricia¹²³⁴⁵

Affiliation:

1. Université Paris Descartes

2. UMR 8601 CNRS

3. Laboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques

4. 75006 Paris

5. France

Abstract

The obtention of 4-amino-3-cyano-N-arylpyrazoles via a μW mediated cyclization allowed the diversity oriented syntheses of various heteroyclic scaffolds.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/OB/C4OB01951B

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